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PI3Kδ inhibitor 52
CAS No. 1911564-39-0
PI3Kδ inhibitor 52 ( —— )
Catalog No. M12995 CAS No. 1911564-39-0
A potent, selective, and efficacious PI3Kδ inhibitor with IC50 of 1.7 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 222 | Get Quote |
|
| 10MG | 357 | Get Quote |
|
| 25MG | 597 | Get Quote |
|
| 50MG | 851 | Get Quote |
|
| 100MG | 1152 | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NamePI3Kδ inhibitor 52
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NoteResearch use only, not for human use.
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Brief DescriptionA potent, selective, and efficacious PI3Kδ inhibitor with IC50 of 1.7 nM.
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DescriptionA potent, selective, and efficacious PI3Kδ inhibitor with IC50 of 1.7 nM, >100-fold selectivitity over PI3Kγ/α/β; shows potent activity in mouse arthritis models.
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Synonyms——
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PathwayPI3K/Akt/mTOR signaling
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TargetPI3K
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RecptorPI3K
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Research AreaInflammation/Immunology
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Indication——
Chemical Information
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CAS Number1911564-39-0
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Formula Weight471.44
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Molecular FormulaC22H20F3N7O2
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Purity>98% (HPLC)
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Solubility——
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SMILESCC(=O)N1CCN(C(=O)C1(C)C)C2=C(C=CC(=C2)C3=CC(=C4N3N=CN=C4N)C(F)(F)F)C#N
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Chemical Name2-(4-acetyl-3,3-dimethyl-2-oxopiperazin-1-yl)-4-(4-amino-5-(trifluoromethyl)pyrrolo[2,1-f][1,2,4]triazin-7-yl)benzonitrile
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Liu Q, et al. J Med Chem. 2017 Jun 22;60(12):5193-5208.
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